Clobenpropit (dihydrobromide), CAS [[145231-35-2]]

Artikelnummer: MCE-HY-101198
Artikelname: Clobenpropit (dihydrobromide), CAS [[145231-35-2]]
Artikelnummer: MCE-HY-101198
Hersteller Artikelnummer: HY-101198
Alternativnummer: MCE-HY-101198-25MG,MCE-HY-101198-5MG,MCE-HY-101198-50MG,MCE-HY-101198-10MG,MCE-HY-101198-100MG,MCE-HY-101198-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Clobenpropit dihydrobromide is a potent histamine H3R antagonist/inverse agonist with a pEC50 of 8.07 for histamine H3LR[1]. Clobenpropit dihydrobromide acts as partial agonist at histamine H4 receptors (Ki 13 nM). Clobenpropit dihydrobromide also binds to serotonin 5-HT3 receptors (Ki 7.4 nM) and alpha2A/alpha2C adrenoceptors (Ki 17.4/7.8 nM)[2]. Clobenpropit dihydrobromide increases apoptosis[3].
Molekulargewicht: 470.65
Reinheit: 99.76
CAS Nummer: [145231-35-2]
Formel: C14H19Br2ClN4S
Target-Kategorie: Apoptosis,Histamine Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound