Lintitript (SR 27897) is a highly potent, selective, orally active, competitive and non-peptide cholecystokinin (CCK1) receptor antagonist with an EC50 of 6 nM and a Ki of 0.2 nM. Lintitript displays > 33-fold selectivity more selective for CCK1 than CCK2 receptors (EC50 value of 200 nM). Lintitript increases plasma concentration of leptin and food intake as well as plasma concentration of insulin[1][2][3].
Molekulargewicht:
411.86
Reinheit:
99.58
CAS Nummer:
[136381-85-6]
Formel:
C20H14ClN3O3S
Target-Kategorie:
Cholecystokinin Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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