Gaboxadol (hydrochloride), CAS [[85118-33-8]]

Artikelnummer: MCE-HY-10233
Artikelname: Gaboxadol (hydrochloride), CAS [[85118-33-8]]
Artikelnummer: MCE-HY-10233
Hersteller Artikelnummer: HY-10233
Alternativnummer: MCE-HY-10233-50MG,MCE-HY-10233-5MG,MCE-HY-10233-100MG,MCE-HY-10233-10MG,MCE-HY-10233-10MMX1ML,MCE-HY-10233-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: Lu 02-030 (hydrochloride), THIP (hydrochloride)
Gaboxadol hydrochloride (Lu 02-030 hydrochloride) is a potent agonist of the GABAA receptor and an antagonist of GABAC receptors (IC50=25 µM). Gaboxadol hydrochloride displays a partial agonist efficacy on subunit alpha1beta2gamma2 with an ED50 value of 143 µM, a full agonist efficacy at alpha5 subunit (ED50=28-129 µM) and a superagonist efficacy at alpha4beta3delta (ED50=6 µM). Gaboxadol hydrochloride is a non-opioid agent[1][2].
Molekulargewicht: 176.60
Reinheit: 99.95
CAS Nummer: [85118-33-8]
Formel: C6H9ClN2O2
Target-Kategorie: GABA Receptor
Anwendungsbeschreibung: Reference compound