8-(3-Chlorostyryl)caffeine, CAS [[148589-13-3]] Preis auf Anfrage

Artikelnummer: MCE-HY-103164A
Artikelname: 8-(3-Chlorostyryl)caffeine, CAS [[148589-13-3]] Preis auf Anfrage
Artikelnummer: MCE-HY-103164A
Hersteller Artikelnummer: HY-103164A
Alternativnummer: MCE-HY-103164A-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: CSC
8-(3-Chlorostyryl)caffeine (CSC) is an adenosine antagonist with selective activity at the A2a adenosine receptor. 8-(3-Chlorostyryl)caffeine showed 520-fold selectivity in radioligand binding experiments in rat brain. Antagonism of adenylylase by 8-(3-Chlorostyryl)caffeine shows 22-fold selectivity in rat chromaffin cells When 8-(3-Chlorostyryl)caffeine is co-administered with the A1-selective antagonist CPX, It can also further increase exercise activity. 8-(3-Chlorostyryl)caffeine exhibits good MAO-B inhibitory activity in primate mitochondria. 8-(3-Chlorostyryl)caffeine also has excellent A2A receptor affinity[1].
Molekulargewicht: 330.77
CAS Nummer: [148589-13-3]
Formel: C16H15ClN4O2
Target-Kategorie: Endogenous Metabolite
Anwendungsbeschreibung: MCE Product type: Reference compound