Fasudil (Hydrochloride) (Standard), CAS [[105628-07-7]]

Artikelnummer: MCE-HY-10341R
Artikelname: Fasudil (Hydrochloride) (Standard), CAS [[105628-07-7]]
Artikelnummer: MCE-HY-10341R
Hersteller Artikelnummer: HY-10341R
Alternativnummer: MCE-HY-10341R-100MG,MCE-HY-10341R-50MG,MCE-HY-10341R-25MG,MCE-HY-10341R-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: HA-1077 (Hydrochloride) (Standard), AT-877 (Hydrochloride) (Standard)
Fasudil (Hydrochloride) (Standard) is the analytical standard of Fasudil (Hydrochloride). This product is intended for research and analytical applications. Fasudil (HA-1077, AT877) Hydrochloride is a nonspecific RhoA/ROCK inhibitor and also has inhibitory effect on protein kinases, with an Ki of 0.33 µM for ROCK1, IC50s of 0.158 µM and 4.58 µM, 12.30 µM, 1.650 µM for ROCK2 and PKA, PKC, PKG, respectively. Fasudil Hydrochloride is also a potent Ca2+ channel antagonist and vasodilator[1][2][3].
Molekulargewicht: 327.83
CAS Nummer: [105628-07-7]
Formel: C14H18ClN3O2S
Target-Kategorie: Autophagy,Calcium Channel,HIV,PKA,PKC,Reference Standards,ROCK
Anwendungsbeschreibung: MCE Product type: Reference Standards