SKF-83566, CAS [[99295-33-7]]

Produktübersicht

• Artikelname: SKF-83566, CAS [[99295-33-7]]
• Artikelnummer: MCE-HY-103430A
• Hersteller Artikelnummer: HY-103430A
• Alternativnummer: MCE-HY-103430A-10MMX1ML,MCE-HY-103430A-25MG,MCE-HY-103430A-5MG,MCE-HY-103430A-10MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

SKF-83566 is a potent, blood-brain permeable and orally active D1-like dopamine receptor (D1DR) antagonist and a weaker competitive antagonist at the vascular 5-HT2 receptor (Ki=11 nM)[1][3]. SKF-83566 is a competitive DAT (dopamine transporter) inhibitor with an IC50 of 5.7 µM[2]. SKF-83566 also shows selective inhibition for adenylyl cyclase 2 (AC2) over AC1 and AC5 in the isolated rabbit thoracic aorta[4]. SKF-83566 can be used for research of parkinsons disease and nicotine craving alleviation[5].

Produkteigenschaften

• Molekulargewicht: 332.23
• Reinheit: 99.86
• CAS Nummer: [99295-33-7]
• Formel: C17H18BrNO
• Target-Kategorie: 5-HT Receptor,Adenylate Cyclase,Dopamine Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound