SA57 is a potent, selective FAAH inhibitor with IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH. SA57 also inhibits the 2-arachidonoylglycerol hydrolases MAGL (IC50s of 410 nM and 1.4 µM for mouse and human MAGL) and mouse alpha/beta-hydrolase domain-containing protein 6 (mABHD6, IC50 of 850 nM), but not other brain serine hydrolases[1][2].
Molekulargewicht:
338.83
Reinheit:
99
CAS Nummer:
[1346169-63-8]
Formel:
C17H23ClN2O3
Target-Kategorie:
FAAH,MAGL
Anwendungsbeschreibung:
MCE Product type: Reference compound
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