THIQ (Standard), CAS [[312637-48-2]] Preis auf Anfrage

Produktübersicht

• Artikelname: THIQ (Standard), CAS [[312637-48-2]] Preis auf Anfrage
• Artikelnummer: MCE-HY-10624R
• Hersteller Artikelnummer: HY-10624R
• Alternativnummer: MCE-HY-10624R-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

THIQ (Standard) is the analytical standard of THIQ (HY-10624). This product is intended for research and analytical applications. THIQ is the first selective agonist of the melanocortin-4 receptor (MC4R), with high affinity and potency for hMC4R (IC50=1.2 nM, EC50=2.1 nM) and rMC4R (IC50=0.6 nM, EC50=2.9 nM). THIQ maintains low potency at MC1R, MC3R and MC5R. THIQ plays a role in eliciting erectile activity in rodents. THIQ acts as a pharmacoperone of the MC4R rescuing the cell surface expression and signaling of some intracellularly retained MC4R mutants[1][2].

Produkteigenschaften

• Molekulargewicht: 589.17
• CAS Nummer: [312637-48-2]
• Formel: C33H41ClN6O2
• Target-Kategorie: Melanocortin Receptor,Reference Standards

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference Standards