Urotensin-II receptor antagonist-1, CAS [[1034708-07-0]] Preis auf Anfrage
Artikelnummer:
MCE-HY-10672
| Artikelname: |
Urotensin-II receptor antagonist-1, CAS [[1034708-07-0]] Preis auf Anfrage |
| Artikelnummer: |
MCE-HY-10672 |
| Hersteller Artikelnummer: |
HY-10672 |
| Alternativnummer: |
MCE-HY-10672-1UNIT |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| Urotensin-II receptor antagonist-1 (compound 1) is a low oral bioavailability (F=0-3%, rat) selective human Urotensin II receptor antagonist, Ki=16 nM (test on HEK293 cells expressing recombinant human UT receptor). Urotensin-II receptor antagonist-1 inhibits cytochrome P450 (IC50=0.75 µM, CYP2D6, 1.4 µM, CYP3A4), inhibits kappa-opioid receptor (EC50=3.2 µM), targets cardiac sodium channels (Ki=2.5 µM)[1]. |
| Molekulargewicht: |
460.44 |
| CAS Nummer: |
[1034708-07-0] |
| Formel: |
C25H31Cl2N3O |
| Target-Kategorie: |
Cytochrome P450,Opioid Receptor,Sodium Channel,Urotensin Receptor |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound1 |
