Amosulalol (YM 09538) is an orally active and dual inhibitor of alpha1/beta1-Adrenergic Receptor. Amosulalol exhibits antihypertensive activity via alpha1-Adrenergic Receptor inhibition. Amosulalol decreases reflexogenic increases in heart rate and plasma renin activity (PRA) via beta1-Adrenergic Receptor inhibition in spontaneously hypertensive rats (SHR)[1].
Molekulargewicht:
380.46
Reinheit:
98.69
CAS Nummer:
[85320-68-9]
Formel:
C18H24N2O5S
Target-Kategorie:
Adrenergic Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound1
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