Epertinib (S-22611) hydrochloride is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR, HER4 and HER2, with IC50s of 1.48 nM, 2.49 nM and 7.15 nM, respectively. Epertinib hydrochloride shows potent antitumor activity[1][2]. Epertinib (hydrochloride) is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
Molekulargewicht:
596.48
Reinheit:
98.15
CAS Nummer:
[2071195-74-7]
Formel:
C30H28Cl2FN5O3
Target-Kategorie:
EGFR
Anwendungsbeschreibung:
MCE Product type: Reference compound
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