SNAP 94847 is a novel, high affinity selective melanin-concentrating hormonereceptor1 (MCHR1) antagonist with (Ki= 2.2 nM, Kd=530 pM), it displays >80-fold and >500-fold selectivity over MCHalpha1A and MCHD2 receptors respectively. SNAP 94847 binds with high affinity to the mouse and rat MCHR1 with minimal cross-reactivity to other GPCR, ion channels, enzymes, and transporters[1][3].
Molekulargewicht:
478.57
CAS Nummer:
[487051-12-7]
Formel:
C29H32F2N2O2
Target-Kategorie:
MCHR1 (GPR24)
Anwendungsbeschreibung:
MCE Product type: Reference compound
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