SNAP 94847 hydrochloride is a novel, high affinity selective melanin-concentrating hormonereceptor1 (MCHR1) antagonist with (Ki= 2.2 nM, Kd=530 pM), it displays >80-fold and >500-fold selectivity over MCHalpha1A and MCHD2 receptors respectively. SNAP 94847 hydrochloride binds with high affinity to the mouse and rat MCHR1 with minimal cross-reactivity to other GPCR, ion channels, enzymes, and transporters[1][3].
Molekulargewicht:
515.03
Reinheit:
99.90
CAS Nummer:
[1781934-47-1]
Formel:
C29H33ClF2N2O2
Target-Kategorie:
MCHR1 (GPR24)
Anwendungsbeschreibung:
MCE Product type: Reference compound
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