SR 142948 (Standard), CAS [[184162-64-9]] Preis auf Anfrage

Artikelnummer: MCE-HY-107664R
Artikelname: SR 142948 (Standard), CAS [[184162-64-9]] Preis auf Anfrage
Artikelnummer: MCE-HY-107664R
Hersteller Artikelnummer: HY-107664R
Alternativnummer: MCE-HY-107664R-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
SR 142948 (Standard) is the analytical standard of SR 142948 (HY-107664). This product is intended for research and analytical applications. SR 142948 is an orally active and selective non-peptide neurotensin receptor (NT) antagonist with IC50s of 1.19 nM, 0.32 nM, 3.96 nM in h-NTR1-CHO cells, HT-29 cells, and adult rat brain, respectively. SR 142948 antagonizes NT-induced inositol monophosphate formation in HT-29 cells with an IC50 of 3.9 nM. SR 142948 blocks hypothermia, analgesia and steering behavior induced by NT in vivo. SR 142948 shows blood-brain permeability and can be used in study of psychiatric disorders[1][2].
Molekulargewicht: 685.85
CAS Nummer: [184162-64-9]
Formel: C39H51N5O6
Target-Kategorie: Neurotensin Receptor,Reference Standards
Anwendungsbeschreibung: MCE Product type: Reference Standards