CGP 78608 hydrochloride is a highly potent and selective antagonist at the glycine-binding site of the NMDA receptor, with an IC50 of 6 nM. CGP 78608 hydrochloride acts as a potentiator of GluN1/GluN3A-mediated glycine currents, with an estimated EC50 in the low nM range (26.3 nM). Anticonvulsant activity[1][2].
Molekulargewicht:
414.58
Reinheit:
99.56
CAS Nummer:
[1135278-54-4]
Formel:
C11H14BrClN3O5P
Target-Kategorie:
iGluR
Anwendungsbeschreibung:
MCE Product type: Reference compound
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