BIX-01294 (trihydrochloride), CAS [[1392399-03-9]]

Artikelnummer: MCE-HY-108239
Artikelname: BIX-01294 (trihydrochloride), CAS [[1392399-03-9]]
Artikelnummer: MCE-HY-108239
Hersteller Artikelnummer: HY-108239
Alternativnummer: MCE-HY-108239-100MG,MCE-HY-108239-250MG,MCE-HY-108239-500MG,MCE-HY-108239-1G,MCE-HY-108239-25MG,MCE-HY-108239-10MG,MCE-HY-108239-5MG,MCE-HY-108239-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
BIX-01294 trihydrochloride is a reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor, with IC50s of of 1.7 µM and 0.9 µM, respectively. BIX-01294 trihydrochloride inhibits G9a/GLP by competing for binding with the amino acids N-terminal of the substrate lysine residue. BIX-01294 trihydrochloride, a (1H-1,4-diazepin-1-yl)-quinazolin-4-yl amine derivative, induces necroptosis and autophagy. BIX-01294 trihydrochloride has antitumor activity in recurrent tumor cells[1][2][3][4][5].
Molekulargewicht: 600.02
Reinheit: 99.68
CAS Nummer: [1392399-03-9]
Formel: C28H41Cl3N6O2
Target-Kategorie: Autophagy,Histone Methyltransferase
Anwendungsbeschreibung: MCE Product type: Reference compound