Lanraplenib succinate (GS-9876 succinate) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases. Lanraplenib succinate (GS-9876 succinate) inhibits SYK activity in platelets via the glycoprotein VI (GPVI) receptor without prolonging bleeding time (BT) in monkeys or humans[1][2][3].
Molekulargewicht:
620.64
Reinheit:
98.09
CAS Nummer:
[1800047-00-0]
Formel:
C23H25N9O.3/2C4H6O4
Target-Kategorie:
Syk
Anwendungsbeschreibung:
MCE Product type: Reference compound
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