Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist with EC50 values of 8.16, 3.91, 1.14 and 0.251 nM for human (h), cynomolgus monkey (cm), mouse (m) and rat (r) MC1R, respectively. Dersimelagon shows good affinity for hMC1R and hMC4R with Ki values of 2.26, 32.9 nM, respectively. Dersimelagon can be used for the research of skin pigmentation[1][2].
Molekulargewicht:
675.75
Reinheit:
98.66
CAS Nummer:
[1835256-48-8]
Formel:
C36H45F4N3O5
Target-Kategorie:
Melanocortin Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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