NF449 (octasodium), CAS [[627034-85-9]]

Artikelnummer: MCE-HY-112461A
Artikelname: NF449 (octasodium), CAS [[627034-85-9]]
Artikelnummer: MCE-HY-112461A
Hersteller Artikelnummer: HY-112461A
Alternativnummer: MCE-HY-112461A-25MG, MCE-HY-112461A-100MG, MCE-HY-112461A-10MG, MCE-HY-112461A-1MG, MCE-HY-112461A-50MG, MCE-HY-112461A-5MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
NF449 octasodium is a highly potent P2X1 receptor antagonist, with IC50s of 0.28, 0.69, and 120 nM for rP2X1, rP2X1+5, P2X2+3, respectively. NF449 octasodium is a Gsalpha-selective G Protein antagonist. NF449 octasodium suppresses the rate of GTP[gammaS] binding to Gsalpha-s, inhibits the stimulation of adenylyl cyclase activity, and blocks the coupling of beta-adrenergic receptors to Gs[1][2].
Molekulargewicht: 1505.09
Reinheit: 99
CAS Nummer: [627034-85-9]
Formel: C41H24N6Na8O29S8
Target-Kategorie: P2X Receptor
Anwendungsbeschreibung: Reference compound