Almonertinib (mesylate), CAS [[2134096-06-1]]

Artikelnummer: MCE-HY-112823A
Artikelname: Almonertinib (mesylate), CAS [[2134096-06-1]]
Artikelnummer: MCE-HY-112823A
Hersteller Artikelnummer: HY-112823A
Alternativnummer: MCE-HY-112823A-100MG,MCE-HY-112823A-10MG,MCE-HY-112823A-50MG,MCE-HY-112823A-5MG,MCE-HY-112823A-25MG,MCE-HY-112823A-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: HS-10296 (mesylate)
Almonertinib (HS-10296) mesylate is an orally available, irreversible, third-generation EGFR tyrosine kinase inhibitor with high selectivity for EGFR-sensitizing and T790M resistance mutations. Almonertinib mesylate shows great inhibitory activity against T790M, T790M/L858R and T790M/Del19 (IC50: 0.37, 0.29 and 0.21 nM, respectively), and is less effective against wild type (3.39 nM). Almonertinib mesylate is used for the research of the non-small cell lung cancer[1][2].
Molekulargewicht: 621.75
Reinheit: 99.67
CAS Nummer: [2134096-06-1]
Formel: C31H39N7O5S
Target-Kategorie: EGFR
Anwendungsbeschreibung: Reference compound