Osavampator (TAK-653) is a AMPA receptor positive allosteric modulator. Osavampator selectively binds to AMPA-R in a glutamate-dependent manner and induces Ca2+ influx in hGluA1i CHO cells (EC50 = 3.3 µM). Osavampator improves learning and memory in many models. Osavampator is can be used for the research of depressive disorders[1][2].
Molekulargewicht:
373.47
Reinheit:
99.74
CAS Nummer:
[1358751-06-0]
Formel:
C19H23N3O3S
Target-Kategorie:
iGluR,Lipoxygenase
Anwendungsbeschreibung:
MCE Product type: Reference compound
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