TSR-011-isomer, CAS [[1388225-79-3]] Preis auf Anfrage

Artikelnummer: MCE-HY-117806
Artikelname: TSR-011-isomer, CAS [[1388225-79-3]] Preis auf Anfrage
Artikelnummer: MCE-HY-117806
Hersteller Artikelnummer: HY-117806
Alternativnummer: MCE-HY-117806-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
TSR-011-isomer is an isomer of Belizatinib (HY-17603), a ALK inhibitor with an IC50 of 6 nM. TSR-011-isomer acts as a substrate for metabolic hydrolysis and NADPH-dependent metabolism. TSR-011-isomer undergoes enzymatic hydrolysis in mouse plasma and NADPH-dependent metabolism in mouse liver microsomes, thereby supporting clearance processes. TSR-011-isomer can be used in studies related to ALK-driven cancers[1].
Molekulargewicht: 595.72
CAS Nummer: [1388225-79-3]
Formel: C33H43F2N5O3
Target-Kategorie: Akt,Drug Isomer,NADPH Oxidase
Anwendungsbeschreibung: MCE Product type: Reference compound