VPC-3033, CAS [[110763-24-1]] Preis auf Anfrage

Artikelnummer: MCE-HY-118409
Artikelname: VPC-3033, CAS [[110763-24-1]] Preis auf Anfrage
Artikelnummer: MCE-HY-118409
Hersteller Artikelnummer: HY-118409
Alternativnummer: MCE-HY-118409-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
VPC-3033 is an androgen receptor antagonist. VPC-3033 has a strong androgen DHT replacement potency (IC50: 0.625-2.5 µM), can effectively inhibit androgen receptor transcriptional activity (IC50=0.3 µM), and has a strong androgen receptor degradation ability. In addition, VPC-3033 exhibits significant anti-androgen receptor activity against prostate cancer cells resistant to Enzalutamide (HY-70002)[1].
Molekulargewicht: 298.33
CAS Nummer: [110763-24-1]
Formel: C21H14O2
Target-Kategorie: Androgen Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound