UCPH-102 is a highly selective EAAT1 inhibitor with an IC50 of 0.43 µM. UCPH-102 exhibits a specific anti-proliferative effect on T-ALL cells. UCPH-102 also shows good blood-brain permeability, which can be used in studies of amyotrophic lateral sclerosis, Alzheimers disease, chronic pain and obsessive compulsive disorder[1][2][3][4].
Molekulargewicht:
330.38
Reinheit:
99.20
CAS Nummer:
[1229591-56-3]
Formel:
C21H18N2O2
Target-Kategorie:
EAAT
Anwendungsbeschreibung:
MCE Product type: Reference compound
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