BMS-599626 (Hydrochloride), CAS [[873837-23-1]]

Artikelnummer: MCE-HY-12010
Artikelname: BMS-599626 (Hydrochloride), CAS [[873837-23-1]]
Artikelnummer: MCE-HY-12010
Hersteller Artikelnummer: HY-12010
Alternativnummer: MCE-HY-12010-100MG,MCE-HY-12010-25MG,MCE-HY-12010-5MG,MCE-HY-12010-10MMX1ML,MCE-HY-12010-10MG,MCE-HY-12010-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: AC480 (Hydrochloride)
BMS-599626 Hydrochloride (AC480 Hydrochloride) is a selective and orally bioavailable HER1 and HER2 inhibitor, with IC50s of 20 and 30 nM, respectively. BMS-599626 Hydrochloride displays ~8-fold less potent to HER4 (IC50=190 nM), >100-fold to VEGFR2, c-Kit, Lck, MEK. BMS-599626 Hydrochloride inhibits tumor cell proliferation, and has potential to increase tumor response to radiotherapy[1][2].
Molekulargewicht: 567.01
Reinheit: 98.90
CAS Nummer: [873837-23-1]
Formel: C27H28ClFN8O3
Target-Kategorie: EGFR
Anwendungsbeschreibung: MCE Product type: Reference compound1