Samelisant (SUVN-G3031) is a potent and selective histamine H3 receptor (H3R) inverse agonist with good brain penetration and oral bioavailability. Samelisant has a similar binding affinity towards human (hH3R, Ki=8.7 nM) and rat (rH3R,Ki=9.8 nM) H3R indicating no inter-species differences. Samelisant can be used for the research of sleep-related disorders[1].
Molekulargewicht:
446.41
Reinheit:
98.65
CAS Nummer:
[1394808-20-8]
Formel:
C21H33Cl2N3O3
Target-Kategorie:
Histamine Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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