2-Bromo-LSD (D-Tartrate), CAS [[2855123-30-5]]

Artikelnummer: MCE-HY-121675A
Artikelname: 2-Bromo-LSD (D-Tartrate), CAS [[2855123-30-5]]
Artikelnummer: MCE-HY-121675A
Hersteller Artikelnummer: HY-121675A
Alternativnummer: MCE-HY-121675A-5MG,MCE-HY-121675A-10MG,MCE-HY-121675A-1MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: BOL-148 (D-Tartrate), Bromolysergide (D-Tartrate)
2-Bromo-LSD D-Tartrate (BOL-148 D-Tartrate) is a blood-brain barrier-permeable 5-HT2A partial agonist and competitive partial antagonist. 2-Bromo-LSD D-Tartrate acts as both a potent partial agonist (with an EC50 of 0.81 nM for Gq dissociation) and a potent partial antagonist (with a KB of 0.18 nM for Gq dissociation) at the 5-HT2A receptor. 2-Bromo-LSD D-Tartrate exhibits partial agonist activity at multiple aminergic GPCRs, including 5-HT2A. 2-Bromo-LSD D-Tartrate lacks 5-HT2B agonist activity. 2-Bromo-LSD D-Tartrate induces dendritogenesis and spinogenesis. 2-Bromo-LSD D-Tartrate reverses the behavioral effects of chronic stress and increases active coping behaviors in mice[1][2].
Molekulargewicht: 477.39
Reinheit: 99.91
CAS Nummer: [2855123-30-5]
Formel: C20H24BrN3O1/2C4H6O6
Target-Kategorie: 5-HT Receptor,G protein-coupled Bile Acid Receptor 1
Anwendungsbeschreibung: MCE Product type: Reference compound