JNJ-55308942, CAS [[2166558-11-6]]
Artikelnummer:
MCE-HY-123857
| Artikelname: |
JNJ-55308942, CAS [[2166558-11-6]] |
| Artikelnummer: |
MCE-HY-123857 |
| Hersteller Artikelnummer: |
HY-123857 |
| Alternativnummer: |
MCE-HY-123857-25MG,MCE-HY-123857-100MG,MCE-HY-123857-5MG,MCE-HY-123857-10MG,MCE-HY-123857-50MG,MCE-HY-123857-10MMX1ML |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| JNJ-55308942 is a high-affinity, selective, brain-penetrant P2X7 functional antagonist (hP2X7: IC50=10 nM, Ki=7.1 nM, rP2X7: IC50=15 nM, Ki=2.9 nM). JNJ-55308942 is orally bioavailable, binds to brain P2X7 and blocks IL-1beta release from adult rodent brain[1][2]. |
| Molekulargewicht: |
425.32 |
| Reinheit: |
99.92 |
| CAS Nummer: |
[2166558-11-6] |
| Formel: |
C17H12F5N7O |
| Target-Kategorie: |
P2X Receptor |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound |