KW-2581 is a steroidal selective steroid sulfatase inhibitor with an IC50 of 4 nM. KW-2581 inhibits sulfated-estrogen dependent growth of breast cancer cells both in vitro and in vivo. KW-2581 induced regression in E1S-induced tumor growth. KW-2581 can be studied in research on hormone receptors-positive breast cancer[1].
Molekulargewicht:
460.63
CAS Nummer:
[284045-56-3]
Formel:
C25H36N2O4S
Target-Kategorie:
Steroid Sulfatase
Anwendungsbeschreibung:
MCE Product type: Reference compound
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