MK-4541 is an orally active and selective androgen receptor (AR) modulator. MK-4541 acts as an antagonist to inhibit 5alpha-reductase. MK-4541 inhibits proliferation and induces apoptosis in AR positive prostate cancer cells. MK-4541 significantly inhibited the growth of R3327-G prostate tumors in xenograft mouse model[1].
Molekulargewicht:
428.49
CAS Nummer:
[796885-38-6]
Formel:
C22H31F3N2O3
Target-Kategorie:
5 alpha Reductase,Androgen Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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