U-99194 (maleate), CAS [[234757-41-6]]

Artikelnummer: MCE-HY-12701A
Artikelname: U-99194 (maleate), CAS [[234757-41-6]]
Artikelnummer: MCE-HY-12701A
Hersteller Artikelnummer: HY-12701A
Alternativnummer: MCE-HY-12701A-5MG,MCE-HY-12701A-10MG,MCE-HY-12701A-25MG,MCE-HY-12701A-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: U-99194A, PNU-99194A (maleate), JPC-211 (maleate)
U-99194 (PNU-99194) maleate is a selective, potent dopamine D3 receptor antagonist (Ki =160 nM). U-99194 maleate inhibits the activation of D3 receptor mediated by endogenously released dopamine or exogenous D3 agonists. U-99194 maleate abrogates the IPSC-suppressive effect of the D3 agonist PD 128907 in rat hippocampal slices. U-99194 maleate significantly suppresses Nicotine (HY-127019)-induced tremor in mice. U-99194 maleate can be used for the study of dopamine D3 receptor-mediated motor disorders, particularly kinetic tremors[1][2].
Molekulargewicht: 393.47
Reinheit: 99.23
CAS Nummer: [234757-41-6]
Formel: C21H31NO6
Target-Kategorie: Dopamine Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound