FGTI-2734 (mesylate), CAS [[2702297-24-1]]

Artikelnummer: MCE-HY-128350A
Artikelname: FGTI-2734 (mesylate), CAS [[2702297-24-1]]
Artikelnummer: MCE-HY-128350A
Hersteller Artikelnummer: HY-128350A
Alternativnummer: MCE-HY-128350A-10MG,MCE-HY-128350A-25MG,MCE-HY-128350A-10MMX1ML,MCE-HY-128350A-5MG,MCE-HY-128350A-50MG,MCE-HY-128350A-100MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
FGTI-2734 mesylate is a RAS C-terminal mimetic dual farnesyl transferase (FT) and geranylgeranyl transferase-1 (GGT) inhibitor with IC50s of 250 nM and 520 nM for FT and GGT, respectively. FGTI-2734 mesylate can prevent membrane localization of KRAS, hence solving KRAS resistance problem and thwarting mutant KRAS patient-derived pancreatic tumors[1].
Molekulargewicht: 606.73
Reinheit: 99.65
CAS Nummer: [2702297-24-1]
Formel: C27H35FN6O5S2
Target-Kategorie: Farnesyl Transferase,gamma-Glutamyl Transferase (GGT)
Anwendungsbeschreibung: MCE Product type: Reference compound