Eliprodil, CAS [[119431-25-3]]

Produktübersicht

• Artikelname: Eliprodil, CAS [[119431-25-3]]
• Artikelnummer: MCE-HY-12881
• Hersteller Artikelnummer: HY-12881
• Alternativnummer: MCE-HY-12881-50MG,MCE-HY-12881-5MG,MCE-HY-12881-100MG,MCE-HY-12881-10MG,MCE-HY-12881-10MMX1ML,MCE-HY-12881-25MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: SL-820715

Produktbeschreibung

Eliprodil(SL-820715) is a non-competitive NR2B-NMDA receptor antagonist(IC50=1 uM), less potent for NR2A- and NR2C-containing receptors(IC50> 100 uM). IC50 value: Target: NR2B-NMDA antagonist Human N-type Ca2+ channel currents were inhibited by ifenprodil and eliprodil with IC50 values of 50 microM and 10 microM respectively whereas P-type Ca2+ channel currents were inhibited reversibly by ifenprodil and eliprodil with approximate IC50 values of 60 microM and 9 microM respectively. eliprodil (1 microm) produced a moderate reverse rate-dependent prolongation of the action potential duration (7.4+/-1.5, 8.9+/-2.1 and 9.9+/-1.8% at cycle lengths of 300, 1000 and 5000 ms, respectively, n=9).

Produkteigenschaften

• Molekulargewicht: 347.85
• Reinheit: 99.65
• CAS Nummer: [119431-25-3]
• Formel: C20H23ClFNO
• Target-Kategorie: iGluR

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound