VP3.15 (dihydrobromide), CAS [[1281681-33-1]]

Artikelnummer: MCE-HY-128879A
Artikelname: VP3.15 (dihydrobromide), CAS [[1281681-33-1]]
Artikelnummer: MCE-HY-128879A
Hersteller Artikelnummer: HY-128879A
Alternativnummer: MCE-HY-128879A-10MMX1ML,MCE-HY-128879A-25MG,MCE-HY-128879A-100MG,MCE-HY-128879A-5MG,MCE-HY-128879A-10MG,MCE-HY-128879A-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE)7- glycogen synthase kinase (GSK)3 inhibitor, with IC50s of 1.59 µM and 0.88 µM for PDE7 and GSK-3, respectively. VP3.15 dihydrobromide has neuroprotective and neuroreparative activities, thus as potential combined anti-inflammatory and pro-remyelinating therapies for multiple sclerosis (MS)[1].
Molekulargewicht: 528.30
Reinheit: 98.01
CAS Nummer: [1281681-33-1]
Formel: C20H24Br2N4OS
Target-Kategorie: GSK-3,Phosphodiesterase (PDE)
Anwendungsbeschreibung: Reference compound