YM-44781 (free acid), CAS [[173943-29-8]] Preis auf Anfrage
Artikelnummer:
MCE-HY-129296
Hersteller Artikelnummer:
HY-129296
Alternativnummer:
MCE-HY-129296-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
YM-44781 free acid is a non-peptide neuropeptide receptor antagonist with efficient NK(2) and NK(1) receptor antagonist activity. YM-44781 exhibits significant binding affinity on the NK(2) receptor (pKi = 9.94) and also on the NK(1) receptor Higher binding affinity (pKi = 9.09). In addition, YM-44781 also showed significant inhibitory effects on bladder contraction induced by selective NK(1) receptor agonists[1].
Molekulargewicht:
568.51
CAS Nummer:
[173943-29-8]
Formel:
C31H32Cl2FN3O2
Target-Kategorie:
Endogenous Metabolite
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten