NMDA-IN-1 (dihydrochloride), CAS [[1784252-90-9]] Preis auf Anfrage

Produktübersicht

• Artikelname: NMDA-IN-1 (dihydrochloride), CAS [[1784252-90-9]] Preis auf Anfrage
• Artikelnummer: MCE-HY-12962A
• Hersteller Artikelnummer: HY-12962A
• Alternativnummer: MCE-HY-12962A-1MG,MCE-HY-12962A-5MG,MCE-HY-12962A-10MG,MCE-HY-12962A-25MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

NMDA-IN-1 dihydrochloride is a selective NMDA NR2B antagonist with a Ki of 0.85 nM, NR2B Ca2+ influx IC50 is 9.7 nM. NMDA-IN-1 dihydrochloride inhibits Glu/Gly stimulated Ca2+ flux in Ltk- cells expressing the hNR1a/NR2B with a IC50 of 9.7 nM. NMDA-IN-1 dihydrochloride has no activities on NR2A, NR2C, NR2D, hERG-channel and alpha1-adrenergic receptor. NMDA-IN-1 dihydrochloride shows excellent activity in the mechanical hyperalgesia assay in rats. NMDA-IN-1 dihydrochloride can be used for the studies of stroke, parkinson, and neuropathic pain[1].

Produkteigenschaften

• Molekulargewicht: 412.33
• CAS Nummer: [1784252-90-9]
• Formel: C20H24Cl2FN3O
• Target-Kategorie: iGluR

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound