NF-56-EJ40 is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM[1].
Molekulargewicht:
443.54
Reinheit:
99.92
CAS Nummer:
[2380230-73-7]
Formel:
C27H29N3O3
Target-Kategorie:
Succinate Receptor 1
Anwendungsbeschreibung:
MCE Product type: Reference compound
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