ARCC-4, CAS [[1973403-00-7]]

Artikelnummer: MCE-HY-130492
Artikelname: ARCC-4, CAS [[1973403-00-7]]
Artikelnummer: MCE-HY-130492
Hersteller Artikelnummer: HY-130492
Alternativnummer: MCE-HY-130492-5MG,MCE-HY-130492-25MG,MCE-HY-130492-10MMX1ML,MCE-HY-130492-10MG,MCE-HY-130492-100MG,MCE-HY-130492-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
ARCC-4 is a low-nanomolar Androgen Receptor (AR) degrader based on PROTAC, with a DC50 of 5 nM. ARCC-4 is an enzalutamide-based von Hippel-Lindau (VHL)-recruiting AR PROTAC and outperforms enzalutamide. ARCC-4 effectively degrades clinically relevant AR mutants associated with antiandrogen therapy[1].
Molekulargewicht: 1024.18
Reinheit: 99.88
CAS Nummer: [1973403-00-7]
Formel: C53H56F3N7O7S2
Target-Kategorie: Androgen Receptor,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound