K-Ras ligand-Linker Conjugate 5, CAS [[2378261-85-7]]

Artikelnummer: MCE-HY-130823
Artikelname: K-Ras ligand-Linker Conjugate 5, CAS [[2378261-85-7]]
Artikelnummer: MCE-HY-130823
Hersteller Artikelnummer: HY-130823
Alternativnummer: MCE-HY-130823-10MG,MCE-HY-130823-100MG,MCE-HY-130823-10MMX1ML,MCE-HY-130823-5MG,MCE-HY-130823-25MG,MCE-HY-130823-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
K-Ras ligand-Linker Conjugate 5 incorporates a ligand for K-Ras recruiting moiety, and a PROTAC linker, which recruit E3 ligases (such as VHL, CRBN, MDM2, and IAP). K-Ras ligand-Linker Conjugate 5 can be used in the synthesis of PROTAC K-Ras Degrader-1 (HY-129523), which is potent PROTAC K-Ras degrader that exhibits 70% degradation efficacy in SW1573 cells[1].
Molekulargewicht: 789.96
Reinheit: 99.79
CAS Nummer: [2378261-85-7]
Formel: C42H59N7O8
Target-Kategorie: Target Protein Ligand-Linker Conjugates
Anwendungsbeschreibung: MCE Product type: Reference compound