K-Ras ligand-Linker Conjugate 6 (formate)

Artikelnummer: MCE-HY-130991A
Artikelname: K-Ras ligand-Linker Conjugate 6 (formate)
Artikelnummer: MCE-HY-130991A
Hersteller Artikelnummer: HY-130991A
Alternativnummer: MCE-HY-130991A-25MG,MCE-HY-130991A-50MG,MCE-HY-130991A-10MG,MCE-HY-130991A-100MG,MCE-HY-130991A-5MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
K-Ras ligand-Linker Conjugate 6 formate incorporates a ligand for K-Ras recruiting moiety, and a PROTAC linker, which recruit E3 ligases (such as VHL, CRBN, MDM2, and IAP). K-Ras ligand-Linker Conjugate 6 formate can be used in the synthesis of PROTAC K-Ras Degrader-1 (HY-129523), which is potent PROTAC K-Ras degrader that exhibits 70% degradation efficacy in SW1573 cells[1].
Molekulargewicht: 835.00
Reinheit: 98.93
Formel: C43H62N8O9
Target-Kategorie: Target Protein Ligand-Linker Conjugates
Anwendungsbeschreibung: Reference compound