LY2934747 is a selective and blood-brain barrier-permeable dual mGlu2/mGlu3 receptor agonist, with Ki values of 260 nM and 177 nM, and EC50 values of 8.4 nM and 62.4 nM against human receptors, respectively. LY2934747 exhibits antipsychotic and analgesic activities in in vivo animal models. LY2934747 can be used in studies related to psychosis and pain[1].
Molekulargewicht:
211.22
CAS Nummer:
[1448707-43-4]
Formel:
C10H13NO4
Target-Kategorie:
mGluR
Anwendungsbeschreibung:
MCE Product type: Reference compound
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