GSK215, CAS [[2743427-26-9]]

Produktübersicht

• Artikelname: GSK215, CAS [[2743427-26-9]]
• Artikelnummer: MCE-HY-132296
• Hersteller Artikelnummer: HY-132296
• Alternativnummer: MCE-HY-132296-10MG,MCE-HY-132296-5MG,MCE-HY-132296-25MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

GSK215 is a potent and selective PROTAC focal adhesion kinase (FAK) degrader with a pDC50 of 8.4. GSK215 is designed by a binder for the VHL E3 ligase and the FAK inhibitor VS-4718. GSK215 induces rapid and prolonged FAK degradation, giving a long-lasting effect on FAK levels and a marked pharmacokinetic/pharmacodynamics (PK/PD) disconnect[1].

Produkteigenschaften

• Molekulargewicht: 985.13
• Reinheit: 99.26
• CAS Nummer: [2743427-26-9]
• Formel: C50H59F3N10O6S
• Target-Kategorie: FAK,PROTACs

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound