RJW103 is an acid-stable SF-1 (NR5A1) and LRH-1 agonist with pEC50 values of 6.5 and 5.9, respectively. RJW103 activates SF-1- and LRH-1-mediated transcription of endogenous target genes. RJW103 can be used in research on cancer, endocrinology and metabolic diseases, such as adrenocortical tumors[1][2].
Molekulargewicht:
385.58
Reinheit:
98.71
CAS Nummer:
[1276664-14-2]
Formel:
C28H35N
Target-Kategorie:
Orphan Nuclear Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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