BM-531 is a dual-acting agent for thromboxane receptor (TXA2) antagonism and thromboxane synthase inhibition. BM-531 exerts anti-aggregatory effects on human citrated platelet-rich plasma (PRP), inhibiting Arachidonic acid (HY-109590A)-induced aggregation with an ED100 of 0.125 µM and U-46619 (HY-108566)-induced aggregation with an ED50 of 0.482 µM. BM-531 inhibits high-K+-induced contraction of porcine uterine smooth muscle[1][2][3].
Molekulargewicht:
398.48
CAS Nummer:
[284464-46-6]
Formel:
C17H26N4O5S
Target-Kategorie:
Prostaglandin Receptor
Anwendungsbeschreibung:
MCE Product type: Biochemical Assay Reagents
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