Raloxifene 4-glucuronide-d4, CAS [[1279033-52-1]] Preis auf Anfrage
Artikelnummer:
MCE-HY-135582S
Hersteller Artikelnummer:
HY-135582S
Alternativnummer:
MCE-HY-135582S-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Raloxifene 4-glucuronide-d4 is deuterated labeled Raloxifene 4-glucuronide (HY-135582). Raloxifene 4-glucuronide is a primary metabolite of Raloxifene. Raloxifene 4-glucuronide formation is mediated mostly by UGT1A10 and UGT1A8. Raloxifene 4-glucuronide binds to estrogen receptor with an IC50 of 370 µM. [1][2]. Raloxifene is a selective estrogen receptor modulator. Raloxifene activates TGFbeta3 promoter as a full agonist at nanomolar concentrations, and inhibits the estrogen response element-containing vitellogenin promoter expression[3].
Molekulargewicht:
653.73
CAS Nummer:
[1279033-52-1]
Formel:
C34H31D4NO10S
Target-Kategorie:
Estrogen Receptor/ERR,Isotope-Labeled Compounds
Anwendungsbeschreibung:
MCE Product type: Isotope-Labeled Compounds
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