GPR81 agonist 1 is a potent and highly selective GPR81 agonist, with EC50s of 58 nM and 50 nM for human and mouse GPR81, respectively. GPR81 agonist 1 inhibits lipolysis in differentiated 3T3-L1 adipocytes. GPR81 agonist 1 suppresses lipolysis in mice without cutaneous flushing. GPR81 agonist 1 displays remarkable selectivity for GPR81 over GPR109a[1].
Molekulargewicht:
446.63
Reinheit:
99.73
CAS Nummer:
[1620992-67-7]
Formel:
C22H30N4O2S2
Target-Kategorie:
Hydroxycarboxylic Acid Receptor (HCAR)
Anwendungsbeschreibung:
MCE Product type: Reference compound
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