GRK5-IN-2 (compound 707), a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor with an IC50 of 49.7 µM. GRK5-IN-2 regulates the expression and/or release of insulin and is useful for the metabolic disease research[1][2].
Molekulargewicht:
380.40
Reinheit:
99.91
CAS Nummer:
[1642839-27-7]
Formel:
C20H20N4O4
Target-Kategorie:
ERK,G Protein-coupled Receptor Kinase (GRK)
Anwendungsbeschreibung:
MCE Product type: Reference compound
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