LSD1-IN-16 (compound 4b) is a potent LSD1 inhibitor. LSD1-IN-16 can inhibit LSD1-CoREST, MAO-A and MAO-B, with IC50 values of 0.015, 0.024, and 0.366 µM, respectively. LSD1-IN-16 displays cell growth arrest in prostate cancer LNCaP cells, with an IC50 of 15.2 µM[1].
Molekulargewicht:
334.43
Formel:
C20H18N2OS
Target-Kategorie:
Histone Demethylase,Monoamine Oxidase
Anwendungsbeschreibung:
MCE Product type: Reference compound
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