NRX-1933 is a type of molecular glue. NRX-1933 is a beta-catenin:beta-TrCP interaction enhancer for the development of small molecule degraders. NRX-1933 promotes the ubiquitination of mutated beta-Catenin, leading to degradation. NRX-1933 can be applied to tumor research on abnormal activation of Wnt/beta - catenin signaling pathway[1][2].
Molekulargewicht:
350.26
Reinheit:
99.51
CAS Nummer:
[2763260-30-4]
Formel:
C14H9F3N6O2
Target-Kategorie:
Molecular Glues,beta-catenin
Anwendungsbeschreibung:
MCE Product type: Reference compound
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