Ar-V7-IN-1 is a potent inhibitor of Ar-V7. Ar-V7-IN-1 inhibits the transcriptional activity of androgen receptor (AR) and the secretion of prostate-specific antigen (PSA) with an eGFP IC50 of 1232 nM and the PSA IC50 of 1391 µM. Ar-V7-IN-1 has the potential for the research of various indications, in particular cancers such as prostate cancer[1].
Molekulargewicht:
394.09
Reinheit:
98.02
CAS Nummer:
[2230880-25-6]
Formel:
C10H10Br2N4OS
Target-Kategorie:
Androgen Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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